Molecular Formula | C17H21N3O2 |
Molar Mass | 299.37 |
Solubility | DMSO: ≥ 34 mg/mL |
Storage Condition | Keep in dark place,Inert atmosphere,2-8°C |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 3.34 ml | 16.702 ml | 33.404 ml |
5 mM | 0.668 ml | 3.34 ml | 6.681 ml |
10 mM | 0.334 ml | 1.67 ml | 3.34 ml |
5 mM | 0.067 ml | 0.334 ml | 0.668 ml |
biological activity | U93631 is a highly effective ligand of GABAA receptor, its IC50 is 100 nM, GABA induces whole cell Cl flow through recombinant GABAA receptor, this effect will be rapidly inhibited by U93961, and this inhibitory effect decays with time. |